1427743-97-2Relevant academic research and scientific papers
Synthesis, receptor binding and activity of iso and azakainoids
Wang, Wentian,Simovic, Dragan D.,Di, Mingping,Fieber, Lynne,Rein, Kathleen S.
supporting information, p. 1949 - 1952 (2013/04/23)
Two syntheses for the production of an unsubstituted azakainoid are described. The 1,3-dipolar cycloaddition of diazomethane with trans-dibenzyl glutaconate yields a 1-pyrazoline, which may be reduced directly to the pyrazolidine. An unexpected trans-cis
