1428768-78-8Relevant articles and documents
Potential CRF1R PET imaging agents: 1-Fluoroalkylsubstituted 5-halo-3-(arylamino)pyrazin-2(1H)-ones
Denhart, Derek J.,Zuev, Dmitry,Ditta, Jonathan L.,Hartz, Richard A.,Ahuja, Vijay T.,Mattson, Ronald J.,Huang, Hong,Mattson, Gail K.,Zueva, Larisa,Nielsen, Julia M.,Kozlowski, Edward S.,Lodge, Nicholas J.,Bronson, Joanne J.,MacOr, John E.
, p. 2052 - 2055 (2013/04/24)
A series of pyrazinones were prepared and evaluated as potential CRF 1R PET imaging agents. Optimization of their CRF1R binding potencies and octanol-phosphate buffer phase distribution coefficients are discussed herein.