1431859-07-2Relevant academic research and scientific papers
Synthesis of [1,2,3]-triazolo[1,5-a][1,4]benzodiazepines via an unprecedented one-pot Cu-catalyzed azidation-cyclization reaction
Hooyberghs, Geert,De Coster, Hendrik,Vachhani, Dipak D.,Ermolat'Ev, Denis S.,Van Der Eycken, Erik V.
, p. 4331 - 4337 (2013)
A novel three-step approach leading to [1,2,3]-triazolo[1,5-a][1,4] benzodiazepines in moderate to good yields has been developed. The key step is an unprecedented one-pot Cu-catalyzed azidation-cyclization reaction of ortho-bromobenzylpropargylamines.
