144037-41-2Relevant academic research and scientific papers
Transition-Metal-Free Alkylation/Arylation of Benzoxazole via Tf2O-Activated-Amide
Niu, Zhi-Jie,Li, Lian-Hua,Liu, Xue-Yuan,Liang, Yong-Min
, p. 5217 - 5222 (2019/11/13)
A transition-metal-free approach to the alkylation/arylation of benzoxazole was developed by employing Tf2O-activated-amide as the alkylating/arylating reagent. The mild reaction conditions, and particularly insensitivity to air and water, further enhance the synthetic potential in pharmaceutical synthesis. (Figure presented.).
The synthesis and the structure-activity relationships of some substituted benzoxazoles, oxazolo(4,5-b)pyridines, benzothiazoles and benzimidazoles as antimicrobial agents
Yalcin,Oren,Sener,Akin,Ucarturk
, p. 401 - 406 (2007/10/02)
The synthesis of a new series of 2,5-disubstituted benzoxazoles 4a-f, 2-substituted oxazolo(4,5-b)pyridines 5a, b, benzothiazoles 6a, b and benzimidazoles 7a, b is described in order to determine their antimicrobial activities and feasible structure-activ
