1476068-51-5Relevant articles and documents
Efficient synthesis of heterocyclic neurotensin receptor ligands by microwave-assisted aminocarbonylation
Lang, Christopher,Gmeiner, Peter
, p. 2474 - 2480 (2013/09/23)
Marking the heterocyclic neurotensin receptor antagonist SR142948A as a lead compound, the development of an efficient and a practical synthetic route to heterocyclic aryl carboxamides is reported. Thus, a highly efficient and flexible access to these carboxamides was elaborated by taking advantage of microwave-assisted aminocarbonylation reaction mediated by Mo(CO)6, Herrmann's palladacycle, [(t-Bu)3PH]BF4, and DBU.