1519954-08-5Relevant academic research and scientific papers
Synthesis of 1-Amino-1H-Indenes via a Sequential Suzuki-Miyaura Coupling/Petasis Condensation Sequence
Jayaram, Vankudoth,Sridhar, Tailor,Sharma, Gangavaram V. M.,Berrée, Fabienne,Carboni, Bertrand
, p. 1803 - 1811 (2017)
An efficient and straightforward synthesis of 1-amino-1H-indenes is reported from 1,2-bis(boronates) via a sequential Suzuki-Miyaura coupling/Petasis cyclization reaction. Starting from the same monoboronic ester intermediates, an intermolecular version of this approach also afforded (Z)-α,β-unsaturated amino esters in moderate to good yields.
Regio- and stereocontrolled access to ?-boronated unsaturated amino esters and derivatives from (z)-alkenyl 1,2-bis(boronates)
Sridhar, Tailor,Berree, Fabienne,Sharma, Gangavaram V. M.,Carboni, Bertrand
, p. 783 - 789 (2014/04/03)
The Borono-Mannich reaction of (Z)-1-alkene-1,2-diboronic esters proceeded regioselectively at the terminal C-B bond to afford (E)-?-boronated unsaturated amino esters in good yields. These compounds were then subjected to Suzuki couplings for the creatio
