155937-32-9Relevant articles and documents
Synthesis and structure-activity relationships of 1-aminophthalazinium salts as GABA(A) receptor antagonists
Colotta,Cecchi,Catarzi,Filacchioni,Galli,Mori
, p. 95 - 105 (2007/10/02)
The synthesis and in vitro GABA(A) activity as GABA(A) antagonists of some 1-aminophthalazinium salts and imidazophthalazines are reported. Structure-activity relationships and a molecular modelling study allowed us to define the features which determine