156205-52-6Relevant articles and documents
Inhibition of the exo-β-d-glucosaminidase CsxA by a glucosamine-configured castanospermine and an amino-australine analogue
Pluvinage, Benjamin,Ghinet, Mariana G.,Brzezinski, Ryszard,Boraston, Alisdair B.,Stubbs, Keith A.
supporting information; experimental part, p. 4169 - 4172 (2009/12/06)
The synthesis of amino-derivatives of castanospermine and australine and their characterisation as inhibitors of the exo-β-d-glucosaminidase CsxA through enzyme kinetics and X-ray structural analysis is described.
A POTENT INHIBITOR OF β-N-ACETYLGLUCOSAMINIDASES: 6-ACETAMIDO-6-DEOXYCASTANOSPERMINE
Liu, Paul S.,Kang, Mohinder S.,Sunkara, Prasad S.
, p. 719 - 720 (2007/10/02)
A facile synthesis of 6-acetamido-6-deoxycastanospermine (4) is described.The target compound inhibits mammalian β-N-acetylglucosaminidases at or below 1 μM.