156760-54-2Relevant academic research and scientific papers
Selective dopamine D-2 autoreceptor agonists with 8-azaindole substructure: Synthesis and theoretical investigations
Gmeiner,Sommer
, p. 435 - 443 (1994)
Starting from the 1,3-dipolar cycloaddition product 6a the peri-fused β-ketoester 7 is prepared. 7 is employed as a key intermediate for the synthesis of the D-2 autoreceptor agonist 5. Two alternative approaches are used for installing the amino function
