157911-66-5Relevant articles and documents
Efficient Pd-catalyzed amination of heteroaryl halides
Charles, Mark D.,Schultz, Phillip,Buchwald, Stephen L.
, p. 3965 - 3968 (2007/10/03)
(Chemical Equation Presented) The Pd-catalyzed amination of a variety of heteroaryl halides has been accomplished by utilizing bulky electron-rich biaryl phosphine ligands. In particular, we report the first couplings of amines with chloro- and bromoindoles bearing a free NH, as well as the first Pd-catalyzed aminations of a 5-halopyrimidine.
Substituted tertiary amino compound or salt thereof
-
, (2008/06/13)
A substituted tertiary amino compound represented by general formula (I) or a pharmaceutically acceptable salt thereof. They have an aromatase inhibiting activity and are useful as a prophylactic and/or therapeutic agent for breast cancer, mastopathy, end