158584-99-7Relevant articles and documents
Metal-free visible light-promoted synthesis of isothiazoles: A catalytic approach for N-S bond formation from iminyl radicals under batch and flow conditions
Alemán, José,Berton, Mateo,Cabrera-Afonso, María Jesús,Cembellín, Sara,Halima-Salem, Adnane,Maestro, M. Carmen,Marzo, Leyre,Miloudi, Abdellah
supporting information, p. 6792 - 6797 (2020/11/09)
A sustainable synthesis of isothiazoles has been developed using an α-amino-oxy acid auxiliary and applying photoredox catalysis. This simple strategy features mild conditions, broad scope and wide functional group tolerance representing a new enviromenta
Discovery of a Potent and Specific M. tuberculosis Leucyl-tRNA Synthetase Inhibitor: (S)-3-(Aminomethyl)-4-chloro-7-(2-hydroxyethoxy)benzo[c][1,2]oxaborol-1(3H)-ol (GSK656)
Li, Xianfeng,Hernandez, Vincent,Rock, Fernando L.,Choi, Wai,Mak, Yvonne S. L.,Mohan, Manisha,Mao, Weimin,Zhou, Yasheen,Easom, Eric E.,Plattner, Jacob J.,Zou, Wuxin,Pérez-Herrán, Esther,Giordano, Ilaria,Mendoza-Losana, Alfonso,Alemparte, Carlos,Rullas, Joaquín,Angulo-Barturen, I?igo,Crouch, Sabrinia,Ortega, Fátima,Barros, David,Alley
, p. 8011 - 8026 (2017/10/18)
There is an urgent need to develop new and safer antitubercular agents that possess a novel mode of action. We synthesized and evaluated a novel series of 3-aminomethyl 4-halogen benzoxaboroles as Mycobacterium tuberculosis (Mtb) leucyl-tRNA synthetase (L
NEW BICYCLIC DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Page/Page column 53, (2017/05/12)
Compounds of formula (I); wherein R1, R2, R3, R4, R5, R6, R7, R8, R14, W, A and n are as defined in the description. Medicaments.
