160726-10-3Relevant articles and documents
Practical Syntheses of a Novel Tricyclic Dipeptide Mimetic Based on a -Azepino Indoline Nucleus: Application to Angiotensin-Converting Enzyme Inhibition
De Lombaert, Stephane,Blanchard, Louis,Stamford, Lisa B.,Sperbeck, Donald M.,Grim, Michael D.,et al.
, p. 7513 - 7516 (1994)
Two stereocontrolled synthetic approaches towards 5-(S)-amino-1,2,4,5,6,7-hexahydro-azepino indole-4-one-2-(S)-carboxylic acid 1, based on intramolecular Friedel-Crafts acylations, are reported.This conformationally restricted tricyclic dipepti