1607449-74-0Relevant academic research and scientific papers
Diamine derivatives as novel small-molecule, potent, and subtype-selective somatostatin SST3 receptor agonists
Li, Derun,Wu, Zhicai,Yu, Yang,Ball, Richard G.,Guo, Liangqin,Sherer, Edward,He, Shuwen,Hong, Qingmei,Lai, Zhong,Qi, Hongbo,Truong, Quang,Yang, David X.,Chicchi, Gary G.,Tsao, Kwei-Lan,Trusca, Dorina,Trujillo, Maria,Pachanski, Michele,Eiermann, George J.,Howard, Andrew D.,Zhou, Yun-Ping,Zhang, Bei B.,Nargund, Ravi P.,Hagmann, William K.
, p. 690 - 695 (2014/07/07)
A novel class of small-molecule, highly potent, and subtype-selective somatostatin SST3 agonists was discovered through modification of a SST3 antagonist. As an example, (1R,2S)-9 demonstrated not only potent in vitro SST3 agonist activity but also in viv
