1609949-22-5Relevant academic research and scientific papers
Synthesis of heterocycles based on rhodium-catalyzed C-H amination
Takahashi, Keisuke,Yamaguchi, Daisuke,Ishihara, Jun,Hatakeyama, Susumi
, p. 133 - 137 (2014)
A new stereoselective approach to substituted pyrrolidines and piperidines is described that involves Du Bois' C-H -amination reaction, Boc-activation of a cyclic sulfamate group, and base-promoted intramolecular cyclization. This methodology can be utilized for the synthesis of tetrahydrofuran and tetrahydrothiophene derivatives. Georg Thieme Verlag Stuttgart · New York.
