1613696-80-2Relevant academic research and scientific papers
BROMODOMAIN INHIBITOR
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Paragraph 0290, (2016/10/31)
The present invention relates to substituted heterocyclic derivative compounds, compositions comprising said compounds, and the use of said compounds and compositions for epigenetic regulation by inhibition of bromodomain-mediated recognition of acetyl lysine regions of proteins, such as histones. Said compositions and methods are useful for the treatment of cancer and neoplastic disease.
