1620066-67-2

Upstream product

• 603-76-9 1-methylindole 
• 1253966-28-7 4-ethyloxy-1-(4-methylbenzenesulfonyl)-1,2,3-triazole 
• 120-72-9 indole 
• 941-55-9 4-toluenesulfonyl azide 
• 1620066-64-9 4-phenoxy-1-tosyl-1H-1,2,3-triazole 

Relevant academic research and scientific papers

Mild aminoacylation of indoles and pyrroles through a three-component reaction with ynol ethers and sulfonyl azides

An effective method for aminoacylation of indoles and pyrroles has been achieved. The transformation involves a multicomponent one-pot cascade reaction between indoles or pyrroles, ynol ethers, and sulfonyl azides, creating four different bonds regioselectively through N-sulfonyltriazole intermediates. The oxo-tryptamines and oxo-pyrroloethanamines are generated in moderate to high yields under mild reaction conditions.