1620108-52-2Relevant academic research and scientific papers
Arylation and heteroarylation of thienylsulfonamides with organotrifluoroborates
Noreen, Mnaza,Rasool, Nasir,El Khatib, Mirna,Molander, Gary A.
, p. 7243 - 7249 (2014/08/18)
A mild, practical protocol has been developed for the Suzuki cross-coupling of unprotected thienylsulfonamides from air- and bench-stable organotrifluoroborates in the absence of a protecting group on the sulfonamide nitrogen. The developed synthetic method can be applied to the preparation of various arylated and heteroarylated thienylsulfonamides under conditions that are tolerant of a broad range of functional groups.
