163618-07-3Relevant articles and documents
Synthesis and structure-activity relationship of new 1,5-dialkyl-1,5- benzodiazepines as cholecystokinin-2 receptor antagonists
Roberts, Karen,Ursini, Antonella,Barnaby, Robert,Cassar, Paolo G.,Corsi, Mauro,Curotto, Giovanni,Donati, Daniele,Feriani, Aldo,Finizia, Gabriella,Marchioro, Carla,Niccolai, Daniela,Oliosi, Beatrice,Polinelli, Stefano,Ratti, Emiliangelo,Reggiani, Angelo,Tedesco, Giovanna,Tranquillini, Maria E.,Trist, David G.,Van Amsterdam, Franciscus T.M.
, p. 4257 - 4273 (2011/08/21)
This article deals with the synthesis and the activities of some 1,5-dialkyl-3-arylureido-1,5-benzodiazepin-2,4-diones which were prepared as potential CCK2 antagonists, with the intention to find a possible follow up of our lead compound GV150013, showin