168272-92-2Relevant academic research and scientific papers
Novel pyrazole-3-carboxamide derivatives as cannabinoid-1 (CB1) antagonists: Journey from non-polar to polar amides
Sasmal, Pradip K.,Reddy, D. Srinivasa,Talwar, Rashmi,Venkatesham,Balasubrahmanyam,Kannan,Srinivas,Kumar, K. Shiva,Devi, B. Neelima,Jadhav, Vikram P.,Khan, Sanjoy K.,Mohan, Priya,Chaudhury, Hira,Bhuniya, Debnath,Iqbal, Javed,Chakrabarti, Ranjan
scheme or table, p. 562 - 568 (2011/02/25)
The synthesis and biological evaluation of novel pyrazole-3-carboxamide derivatives as CB1 antagonists are described. As a part of eastern amide SAR, various chemically diverse motifs were introduced. In general, a range of modifications were well tolerat
Imidazol-4-one and Imidazole-4-thione Compounds
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Page/Page column 14, (2010/05/13)
Imidazol-4-one or imidazole-4-thione compounds of formula (I): wherein X, R1, R2, R3, R4, R5, and R6 are defined herein. Also disclosed is a method for treating a cannabinoid receptor-mediated disorder with these compounds.
Pyrazole-3-carboxamide derivatives, process for their preparation and pharmaceutical compositions in which they are present
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, (2008/06/13)
The present invention relates to novel pyrazole-3-carboxamide derivatives of the formula STR1 in which the substituents are as defined in the specification. The present invention further relates to a process for the preparation of these novel derivatives and to the pharmaceutical compositions in which they are present.
