17833-87-3Relevant academic research and scientific papers
Studies on synthesis of novel triazole tagged pyrazole fused naphthalene 5-thiazine-5,5-dioxide derivatives, their antimicrobial, and antioxidant activity
Malla Reddy,Nagender,Naresh Kumar,Ahn,Pranay Kumar,Kanugula,Rama Krishna,Kotamraju,Narsaiah
, p. E42-E49 (2014/11/08)
A series of novel triazole tagged pyrazole fused naphthalene-5-thiazine-5, 5-dioxide derivatives 8 and 9 were synthesized starting from sodium salt of saccharin 1. The structure of each intermediate and products was established on the basis of spectroscop
Synthesis, molecular docking and antiviral screening of novel N'-substitutedbenzylidene-2-(4-methyl-5,5-dioxido-3-phenylbenzo[e]pyrazolo[4, 3-c][1,2]thiazin-1(4H)-yl)acetohydrazides
Aslam, Sana,Ahmad, Matloob,Athar, Muhammad Makshoof,Ashfaq, Usman Ali,Gardiner, John M.,Montero, Catherine,Detorio, Mervi,Parvez, Masood,Schinazi, Raymond F.
, p. 2930 - 2946 (2014/05/06)
N'-Substitutedbenzylidene-2-(4-methyl-5,5-dioxido-3-phenylbenzo[e] pyrazolo[4,3-c][1,2]thiazin-1(4H)-yl)acetohydrazides (7a-u) were synthesized through a multistep reaction. The final compounds were screened for anti-HIV-1 and cytotoxic activities. Among
Novel structural hybrids of pyrazolobenzothiazines with benzimidazoles as cholinesterase inhibitors
Aslam, Sana,Zaib, Sumera,Ahmad, Matloob,Gardiner, John M.,Ahmad, Aqeel,Hameed, Abdul,Furtmann, Norbert,Gütschow, Michael,Bajorath, Jürgen,Iqbal, Jamshed
, p. 106 - 117 (2014/04/17)
Two series of novel pyrazolobenzothiazine-based hybrid compounds were efficiently synthesized starting from saccharin sodium salt. Pyrazolo[4,3-c][1,2]benzothiazine scaffolds were N-arylated by using p-fluorobenzaldehyde, followed by the incorporation of
Synthesis, Structure, and Reactivity to Nucleophiles of 3-Benzylidene- and 3-Ethylidene-2,3-dihydro-1,2-benzothiazin-4-one 1,1-Dioxides
Dalla Croce, Piero,Del Monaco, Demetrio,La Rosa, Concetta
, p. 299 - 302 (2007/10/02)
A new approach to (Z)-3-benzylidene- and 3-ethylidene-2,3-dihydro-2-methyl-1,2-benzothiazin-4-one 1,1-dioxides (4) starting from the corresponding 3-acyl derivatives (1) is described.A hypothesis, based on 13C n.m.r. data, that products (4) may be conside
