180623-75-0Relevant academic research and scientific papers
Beta3-Adrenoreceptor agonists, agonist compositions and methods of using
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Page/Page column 20-21; 37, (2008/06/13)
The invention provides β3-adrenoreceptor agonists, pharmaceutical compositions comprising β3-adrenoreceptor agonist compounds, and methods of using such compounds for stimulating, regulating or modulating metabolism of fats in adipos
Iodinated analogs of trimetoquinol as highly potent and selective β2- adrenoceptor ligands
De Los Angeles, Joseph E.,Nikulin, Victor I.,Shams, Gamal,Konkar, Anish A.,Mehta, Ratna,Feller, Dennis R.,Miller, Duane D.
, p. 3701 - 3711 (2007/10/03)
A series of trimetoquinol (1, TMQ) analogs were designed and synthesized based on the lead compound 2, a diiodinated analog of trimetoquinol which exhibits improved selectivity for β2-versus β1-adrenoceptors (AR). To determine the in
