181524-53-8

Upstream product

• 100-02-7 4-nitro-phenol 
• 2130-96-3 O-benzyl-N-tert-butoxycarbonyl-L-tyrosine 
• 13512-59-9 N-(tert-butyloxycarbonyl)-O-(phenylmethyl)-L-tyrosine 4-nitrophenol ester 

Downstream Products

• 130203-28-0 N-Decanoyl-O-benzyl-L-tyrosine-p-nitrophenol ester 
• 181524-61-8 O-Benzyl-PhTX-343-N-α-N^G,N^G'-tri-Cbz-L-arginine-amide 
• 130203-15-5 Bis(N-butyryl-O-benzyl-L-tyrosine)-spermineamide 
• 130203-25-7 Bis-C₁₀-PhTX-343 
• 132087-55-9 C₄₂H₅₂N₆O₆ 
• 132087-54-8 Heptanoic acid [(S)-1-[3-(4-{3-[(S)-2-heptanoylamino-3-(4-hydroxy-phenyl)-propionylamino]-propylamino}-butylamino)-propylcarbamoyl]-2-(4-hydroxy-phenyl)-ethyl]-amide 
• 130203-41-7 O-Benzyl-PhTX-di-2',3'-N,N-BOC-334 
• 130203-42-8 O-Benzyl-PhTX-4'-N-Cbz-433 
• 130203-24-6 Bis-PhTX-343 
• 130306-91-1 <127I2>PhTX-343-arginine 
• 132087-53-7 (S)-2-Acetylamino-N-[3-(4-{3-[(S)-2-acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-propylamino}-butylamino)-propyl]-3-(4-hydroxy-phenyl)-propionamide 
• 130203-22-4 PhTX-343-L-arginin-amide 
• 126890-98-0 <127I2>PhTX-343-L-lysine 
• 130203-33-7 N-Butyryl-O-benzyl-L-tyrosyl-butyl-thermospermine 

Relevant academic research and scientific papers

Structure-binding relation of philanthotoxins from nicotinic acetylcholine receptor binding assay

Philanthotoxins are noncompetitive inhibitors of the nicotinic acetylcholine receptor and the various glutamate receptors. Analogues carrying photoaffinity labels, fluorine atoms for solid-state NMR studies of ligand/receptor interaction, and large head g

Synthesis of novel and photolabile philanthotoxin analogs: Glutamate receptor antagonists

The synthetic methods for 27 novel and photolabile philanthotoxin analogs are described. Most analogs were synthesized by two general methods with modifications of these methods where necessary.