186519-95-9Relevant academic research and scientific papers
Selective N-alkylation of pyrrolopyrimidines and indoles by 'transfer of activation'
Sobolov, Susan B.,Sun, Jianmin,Cooper, Beth A.
, p. 5685 - 5688 (2007/10/03)
The benzene sulfonyl group is used as a 'transfer of activation' reagent to alkylate selectively the NH of both pyrrolopyrimidines and 5-aminoindoles substituted on thienopyrimidines. A variety of primary and secondary alcohols are utilized as alkylating
