187395-94-4Relevant articles and documents
Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor
Blommaert, Armand G. S.,Dh?tel, Hélène,Ducos, Bertrand,Durieux, Christiane,Goudreau, Nathalie,Bado, André,Garbay, Christiane,Roques, Bernard P.
, p. 647 - 658 (2007/10/03)
New constrained cyclic pseudopeptide cholecystokinin-B (CCK-B) agonists have been designed on the basis of conformational characteristics of the potent and selective CCK-B agonist Boc-Trp-(NMe)Nle-Asp-Phe-NH2 (K(i) = 0.8 nM, selectivity ratio C