190521-52-9Relevant academic research and scientific papers
Search for surrogates: A study of endothelin receptor antagonist structure activity relationships
Raju,Okun, Ilya,Stavros, Fiona,Chan, Ming Fai
, p. 933 - 938 (1997)
The aryloxymethylene group was used as a replacement for an ester or amide bond present in a series of ET(A) selective endothelin antagonists. The effect of such replacement on the binding affinity is described.
