191276-34-3Relevant articles and documents
PROCESSES FOR TAXANE DERIVATIVES AND INTERMEDIATES USEFUL THEREIN
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Page/Page column 29-30, (2008/06/13)
The application provides a process for the preparation of taxane derivatives and intermediates useful in such processes.
TAXANE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
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Page 4; 14-16, (2008/06/13)
The invention discloses an oxazolidine intermediate for the synthesis of 14- beta -hydroxy-1,14-carbonate-baccatines bearing a 13-isoserine substituent, and a process for the preparation thereof.
TAXANE DERIVATIVES FUNCTIONALIZED AT THE 14- POSITION AND A PROCESS FOR THE PREPARATION THEREOF
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Page 42, (2008/06/13)
A general process for the functionalization at the 14- position of 13-ketobaccatin derivatives of formula I to give derivatives of formula II wherein the substituents are as defined in the disclosure. The conversion of compounds of formula II in compounds of formula III, wherein the substituents are as defined in the disclosure, is also described.