19240-26-7Relevant academic research and scientific papers
Development of novel enkephalin analogues that have enhanced opioid activities at both μ and δ opioid receptors
Yeon, Sun Lee,Petrov, Ravil,Park, Chad K.,Ma, Shou-Wu,Davis, Peg,Lai, Josephine,Porreca, Frank,Vardanyan, Ruben,Hruby, Victor J.
, p. 5528 - 5532 (2008/03/13)
Enkephalin analogues with a 4-anilidopiperidine scaffold have been designed and synthesized to achieve therapeutic benefit for the treatment of pain due to mixed μ and δ opioid agonist activities. Ligand 16, in which a Dmt-substituted enkephalin-like stru
Dehydrooligopeptides. IV. Synthesis of Various Types of Dehydrodi- and tripeptides by Fragment Condensation and Base-Catalyzed β-Elimination
Shin, Chung-gi,Yonezawa, Yasuchika,Yamada, Toyofumi
, p. 2825 - 2831 (2007/10/02)
The synthesis of dehydrotripeptides, composed of an α-amino acid and two α-dehydroamino acid (DHA) residues, by the direct coupling of N-protected δ1-dehydrotripeptide with DHA ester and by the β-elimination od δ1-dehydrodipeptide co
