203574-75-8Relevant academic research and scientific papers
A convenient synthesis of 5-substituted 1-[1- (diethoxyphosphoryl)alkyl]-1H-1,2,3-triazoles
Sikora, Dorota,Gajda, Tadeusz
, p. 1215 - 1222 (1998)
5-Substituted 1-[1(diethoxyphosphoryl)alkyl]-1H-1,2,3-triazoles were prepared in good yields (61-83%) via thermal 1,3-dipolar cycloaddition of diethyl 1-azidoalkylphosphonates and 2-oxoalkylidene triphenylphosphoranes.
Cycloaddition reactions of azidomethyl phosphonate with acetylenes and enamines. Synthesis of triazoles
Louerat, Frederic,Bougrin, Khalid,Loupy, Andre,De Retana, Ana M. Ochoa,Pagalday, Jaione,Palacios, Francisco
, p. 161 - 170 (2007/10/03)
β-Functionalized alkyltriazoles can be efficiently prepared under solvent-free conditions, eventually by coupling with microwave activation. Cycloadditions of azides and poorly activated acetylenes or enamines are thus possible with interesting selectivity in the latter case.
