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208706-12-1

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  • (1R,1'S,3'R/1R,1'R,3'S)-L-054,264;N-[(1R)-2-[[[(1S*,3R*)-3-(AMinoMethyl)cyclohexyl]Methyl]aMino]-1-(1H-indol-3-ylMethyl)-2-oxoethyl]spiro[1H-indene-1,4'-piperidine]-1'-carboxaMide

    Cas No: 208706-12-1

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  • Wuxi Morality Chemical Co., Ltd
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208706-12-1 Usage

Description

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 is a selective somatostatin sst2 receptor agonist, which is a compound that specifically targets and activates the somatostatin sst2 receptor. This receptor is often overexpressed in tumors, making it a potential therapeutic target for various applications.

Uses

Used in Pharmaceutical Industry:
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 is used as a therapeutic agent for targeting tumors with overexpressed somatostatin receptors. Its application is based on its ability to selectively activate the somatostatin sst2 receptor, which can be used to study signaling pathways related to the receptor and potentially develop targeted cancer treatments.
Used in Research and Development:
In the field of research and development, (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 serves as a valuable tool for studying the role of somatostatin receptors in various biological processes. By selectively activating the sst2 receptor, researchers can gain insights into the receptor's function and its potential as a therapeutic target for cancer and other diseases.
Used in Drug Delivery Systems:
Similar to gallotannin, (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 can also benefit from novel drug delivery systems to enhance its applications and efficacy against cancer cells. Utilizing carriers such as organic and metallic nanoparticles can improve the delivery, bioavailability, and therapeutic outcomes of this selective somatostatin sst2 receptor agonist.

Biological Activity

Potent and selective somatostatin sst 2 receptor agonist (K i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst 2 , sst 1 , sst 4 , sst 3 and sst 5 receptors respectively).

Check Digit Verification of cas no

The CAS Registry Mumber 208706-12-1 includes 9 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 6 digits, 2,0,8,7,0 and 6 respectively; the second part has 2 digits, 1 and 2 respectively.
Calculate Digit Verification of CAS Registry Number 208706-12:
(8*2)+(7*0)+(6*8)+(5*7)+(4*0)+(3*6)+(2*1)+(1*2)=121
121 % 10 = 1
So 208706-12-1 is a valid CAS Registry Number.

208706-12-1SDS

SAFETY DATA SHEETS

According to Globally Harmonized System of Classification and Labelling of Chemicals (GHS) - Sixth revised edition

Version: 1.0

Creation Date: Aug 13, 2017

Revision Date: Aug 13, 2017

1.Identification

1.1 GHS Product identifier

Product name N-[1-(cyclohexylmethylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl]spiro[indene-1,4'-piperidine]-1'-carboxamide

1.2 Other means of identification

Product number -
Other names -

1.3 Recommended use of the chemical and restrictions on use

Identified uses For industry use only.
Uses advised against no data available

1.4 Supplier's details

1.5 Emergency phone number

Emergency phone number -
Service hours Monday to Friday, 9am-5pm (Standard time zone: UTC/GMT +8 hours).

More Details:208706-12-1 SDS

208706-12-1Downstream Products

208706-12-1Relevant articles and documents

Spiro [1H-indene-1,4'-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst2) agonists [1]

Yang, Lihu,Guo, Liangqin,Pasternak, Alexander,Mosley, Ralph,Rohrer, Susan,Birzin, Elizabeth,Foor, Forrest,Cheng, Kang,Schaeffer, James,Patchett, Arthur A.

, p. 2175 - 2179 (2007/10/03)

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