20951-10-4Relevant academic research and scientific papers
BROMODOMAIN INHIBITORS
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Paragraph 0501; 0502, (2015/04/28)
The present invention relates to substituted heterocyclic derivative compounds, compositions comprising said compounds, and the use of said compounds and compositions for epigenetic regulation by inhibition of bromodomain-mediated recognition of acetyl lysine regions of proteins, such as histones. Said compositions and methods are useful for the treatment of cancer and neoplastic disease.
