211388-38-4Relevant articles and documents
Synthesis of 4-oxazolinephenylboronic acid and heterobiaryl oxazolines via a Suzuki reaction
Ghosh, Samir,Kumar, A.Sanjeev,Mehta,Soundararajan,Sen, Subhabrata
scheme or table, p. 205 - 207 (2009/11/30)
An efficient synthesis of 4-oxazolinephenylboronic acid from 4-bromobenzoic acid is reported. The title compound couples with heteroaryl halides in presence of Pd(PPh3)4 and Na2CO3 in aqueous toluene to give het
Positional isomers and analogs of mazindol as potential inhibitors of the cocaine binding site on the dopamine transporter site
Houlihan, William J.,Boja, John W.,Kopajtic, Theresa A.,Kuhar, Michael J.,Degrado, Sylvia J.,Toledo, Leonel
, p. 77 - 90 (2007/10/03)
A series of compounds, where the keto-tautomeric form of mazindol (2b) was modified by placing the 2-(p-chlorobenzoyl) portion of the molecule in the 3- and 4-positions, substituting the imidazo ring A by a 4,4-dimethyl 1- 2-oxazolo ring, and replacing th
Rational Design and Synthesis of a Highly Effective Transition State Anolog Inhibitor of the RTEM-1 β-Lactamase
Martin, Richard,Bryan Jones, J.
, p. 8399 - 8402 (2007/10/02)
The synthesis of (1R)-1-acetamido-2-(3-carboxyphenyl)ethane boronic acid, a rationally designed transition state anolog competitive inhibitor of the RTEM-1 β-lactamase from Escherichia coli, is reported.Kinetic measurements show that, as designed, it is a
