211686-54-3Relevant academic research and scientific papers
α-Alkylation of (S)-Asparagine with Self-Regeneration of the Stereogenic Center: Enantioselective Synthesis of α-Substituted Aspartic Acids
Juaristi, Eusebio,Lopez-Ruiz, Heraclio,Madrigal, Domingo,Ramirez-Quiros, Yara,Escalante, Jaime
, p. 4706 - 4710 (1998)
A convenient method for the α-alkylation of (S)-asparagine with "self-regeneration of the stereogenic center" is described. The synthetic protocol involves stereoselective conversion of (S)-asparagine into enantiopure imino ether (2S,6S)-9, which is then
