216569-12-9

Upstream product

• 216569-15-2 (5R)-4-Benzyl-5-phenyl[1,3,4]oxadiazinan-2-one 
• 216569-13-0 (2R)-2-(N-Benzylnitrosoamino)-2-phenylethanol 
• 216569-14-1 (2R)-2-(N-Benzylhydrazino)-2-phenylethanol 
• 14231-57-3 (R)-N-benzyl-2-phenylglycinol 
• 927-58-2 4-bromobutyroyl chloride 
• 216569-16-3 (5R)-5-Phenyl[1,3,4]oxadiazinan-2-one 

Relevant academic research and scientific papers

Preparation and diastereoselective functionalization of a new chiral non racemic bicyclic hydrazinolactam

Starting with R-(-)-phenylglycinol, the synthesis of a new bicyclic hydrazinolactam 3 was realized on a multigram scale. The reaction scope of the corresponding enolate with various electrophiles has been studied. Good to excellent diastereoselectivities were obtained.