217172-24-2Relevant academic research and scientific papers
Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers
Ryder, Todd R.,Hu, Lain-Yen,Rafferty, Michael F.,Millerman, Elizabeth,Szoke, Balazs G.,Tarczy-Hornoch, Katalin
, p. 1813 - 1818 (1999)
Selective N-type Voltage Sensitive Calcium Channel (VSCC) blockers have shown utility in several models of stroke and pain. A series of N,N- dialkyldipeptidylamines with potent functional activity at N-type VSCC's has been identified. Multiple parallel sy
Substituted peptidylamine calcium channel blockers
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, (2008/06/13)
PCT No. PCT/US98/10838 Sec. 371 Date Jan. 19, 1999 Sec. 102(e) Date Jan. 19, 1999 PCT Filed May 28, 1998 PCT Pub. No. WO98/54123 PCT Pub. Date Dec. 3, 1998The present invention provides compounds that block calcium channels having the Formula I shown belo
