Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers

DOI: 10.1016/S0960-894X(99)00284-X

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1813 - 1818 (1999)

Update date:2022-08-05

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Authors:

Ryder, Todd R.

Hu, Lain-Yen

Rafferty, Michael F.

Millerman, Elizabeth

Szoke, Balazs G.

Tarczy-Hornoch, Katalin

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Article abstract of DOI:10.1016/S0960-894X(99)00284-X

Selective N-type Voltage Sensitive Calcium Channel (VSCC) blockers have shown utility in several models of stroke and pain. A series of N,N- dialkyldipeptidylamines with potent functional activity at N-type VSCC's has been identified. Multiple parallel sy

Full text of DOI:10.1016/S0960-894X(99)00284-X

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