219834-95-4

Usage

Uses

Used in Pharmaceutical Industry:
4-Methoxynaphthalene-1-boronic acid is used as a building block in organic synthesis for the preparation of various pharmaceuticals. Its unique reactivity allows for the creation of a wide range of bioactive compounds, contributing to the development of new drugs and therapeutic agents.
Used in Agrochemical Industry:
In the agrochemical sector, 4-Methoxynaphthalene-1-boronic acid serves as a key intermediate in the synthesis of various agrochemicals. Its incorporation into these compounds can enhance their effectiveness in pest control and crop protection, thereby supporting agricultural productivity.
Used in Materials Science:
4-Methoxynaphthalene-1-boronic acid is also utilized in materials science for the development of novel materials with specific properties. Its integration into material compositions can lead to advancements in areas such as polymer science, nanotechnology, and the creation of functional materials for various applications.
Overall, the versatility of 4-Methoxynaphthalene-1-boronic acid stems from its chemical properties, making it a crucial component in the synthesis of compounds across different industries, from healthcare to agriculture and materials development.

InChI:InChI=1/C11H11BO3/c1-15-11-7-6-10(12(13)14)8-4-2-3-5-9(8)11/h2-7,13-14H,1H3

Upstream product

• 688-74-4 boric acid tributyl ester 
• 7732-18-5 water 
• 5467-58-3 1-bromo-4-methoxynaphthalene 
• 121-43-7 Trimethyl borate 
• 2216-69-5 1-Methoxynaphthalene 
• 5419-55-6 Triisopropyl borate 

Relevant academic research and scientific papers

Electrochemical Synthesis of Biaryls via Oxidative Intramolecular Coupling of Tetra(hetero)arylborates

We report herein versatile, transition metal-free and additive-free (hetero)aryl-aryl coupling reactions promoted by the oxidative electrocoupling of unsymmetrical tetra(hetero)arylborates (TABs) prepared from ligand-exchange reactions on potassium trifluoroarylborates. Exploiting the power of electrochemical oxidations, this method complements the existing organoboron toolbox. We demonstrate the broad scope, scalability, and robustness of this unconventional catalyst-free transformation, leading to functionalized biaryls and ultimately furnishing drug-like small molecules, as well as late stage derivatization of natural compounds. In addition, the observed selectivity of the oxidative coupling reaction is related to the electronic structure of the TABs through quantum-chemical calculations and experimental investigations.

Material for organic electroluminescence device and organic electroluminescence device using the same

The present invention discloses an organic material is represented by the following formula(A), the organic EL device employing the material as light emitting host or dopant of emitting layer, hole blocking layer(HBL), electron blocking layer(EBL), electron transport layer(ETL) and hole transport layer (HTL) can display good performance. wherein A represents a substituted or unsubstituted fused ring hydrocarbon units with two to three rings, m represents an integer of 0 to 10, G, Rs and R1 to R3 are the same definition as described in the present invention.

CARBOXAMIDE OR SULFONAMIDE SUBSTITUTED THIAZOLES AND RELATED DERIVATIVES AS MODULATORS FOR THE ORPHAN NUCLEAR RECEPTOR ROR[GAMMA]

The invention provides modulators for the orphan nuclear receptor RORy and methods for treating RORy mediated diseases by administering these novel RORy modulators to a human or a mammal in need thereof. Specifically, the present invention provides carboxamide or sulfonamide containing cyclic compounds of Formula (1), (1'), (100), (100'), (200) and (200') and the enantiomers, diastereomers, tautomers, /V-oxides, solvates and pharmaceutically acceptable salts thereof.

QSAR guided synthesis of simplified antiplasmodial analogs of naphthylisoquinoline alkaloids

Naphthylisoquinoline alkaloids have attracted considerable interest because of their intriguing structure, their unique biosynthetic origin, and their biological activities against several pathogens causing tropical diseases. Their promising pharmacologic