220932-71-8Relevant academic research and scientific papers
Modulations of the amide function of the preferential dopamine D3 agonist (R,R)-S32504: Improvements of affinity and selectivity for D3 versus D2 receptors
Peglion, Jean-Louis,Poitevin, Christophe,La Cour, Clotilde Mannoury,Dupuis, Delphine,Millan, Mark J.
, p. 2133 - 2138 (2009)
Starting with the preferential dopamine (DA) D3 agonist S32504, we prepared two series of derivatives of the general formula I-A and I-B, in an effort to improve both potency and selectivity. For the first set of derivatives, where the primary
