22274-91-5Relevant academic research and scientific papers
Sulfonamide derivatives as new potent and selective CB2 cannabinoid receptor agonists
Ohta, Hiroshi,Ishizaka, Tomoko,Yoshinaga, Mitsukane,Morita, Aki,Tomishima, Yasumitsu,Toda, Yoshihisa,Saito, Shuji
, p. 5133 - 5135 (2007)
A novel series of sulfonamide derivatives 3, the CB2 receptor agonists, was synthesized and evaluated for activity against the human CB2 receptor. We first identified sulfonamide 3a, which was obtained by random screening of our in-h
Regioselective alkylation of thiazolylsulfonamides: Direct and efficient synthesis of 3-alkylthiazolidene derivatives
Masuda, Naoyuki,Yamamoto, Osamu,Fujii, Masahiro,Ohgami, Tetsuro,Moritomo, Ayako,Kontani, Toru,Kageyama, Shunji,Ohta, Mitsuaki
, p. 2305 - 2316 (2007/10/03)
Various N-3-alkylated thiazolidenesulfonamide derivatives were efficiently prepared by the direct endo-selective alkylation of thiazolylsulfonamides. The effects of different bases and solvents were investigated, and the NaH-THF combination was found to b
