226066-70-2Relevant academic research and scientific papers
Thermal cyclization of N-trifluoroacetyl enehydrazines under mild conditions: A novel entry into the Fischer indole synthesis
Miyata, Okiko,Kimura, Yasuo,Muroya, Kanami,Hiramatsu, Hajime,Naito, Takeaki
, p. 3601 - 3604 (1999)
An efficient thermal cyclization of N-trifluoroacetyl enehydrazines for the synthesis of indoles is described.
Efficient synthesis of indoles using [3,3]-sigmatropic rearrangement of N-trifluoroacetyl enehydrazines
Miyata, Okiko,Takeda, Norihiko,Kimura, Yasuo,Takemoto, Yoshiji,Tohnai, Norimitsu,Miyata, Mikiji,Naito, Takeaki
, p. 3629 - 3647 (2007/10/03)
[3,3]-Sigmatropic rearrangement of N-trifluoroacetyl enehydrazines provides a novel method for the construction of indoles. N-Trifluoroacetyl enehydrazine having a cyclopentene ring smoothly underwent [3,3]-sigmatropic rearrangement followed by cyclizatio
One-pot synthesis of indoles from ketones and hydrazines under mild reaction conditions
Miyata,Kimura,Naito
, p. 1635 - 1638 (2007/10/03)
A facile one-pot method is presented for the synthesis of indoles via condensation of ketone with hydrazine followed by acylation and rearrangement. This convenient synthetic method provides an easy and simple access to indoles.
