23328-05-4Relevant articles and documents
SYNTHESIS OF 1,4-EPIMINE COMPOUNDS. IODOSOBENZENE DIACETATE, AN EFFICIENT REAGENT FOR NEUTRAL NITROGEN RADICAL GENERATION
Armas, P. de,Carrau, R.,Concepcion, J. I.,Francisco, C. G.,Hernandez, R.,Suarez, E.
, p. 2493 - 2496 (1985)
Photolysis of several nitroamines, cianamines, and phosphoroamidates in the presence of iodosobenzene diacetate (IBDA) and iodine leads to neutral aminyl radicals which undergo intramolecular hydrogen abstraction to produce epimine compounds with yields t
20-triazole-20-hydroxyl-pregnane derivatives, method for preparing same and medical application of 20-triazole-20-hydroxyl-pregnane derivatives
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, (2018/11/22)
The invention belongs to the field of medicines, and particularly relates to a series of 20-triazole-20-hydroxyl-pregnane derivatives, a method for preparing the same and medical application of the 20-triazole-20-hydroxyl-pregnane derivatives. The 20-triazole-20-hydroxyl-pregnane derivatives are particularly used for preparing medicines for treating androgen receptor related diseases such as cellproliferation, prostate cancer, polytrichia, acne and androgenic alopecia which are dependent on androgens. Structural general formulas of compounds of the 20-triazole-20-hydroxyl-pregnane derivativesare shown. Details of definition of various groups in the general formulas are attached to specifications.
Synthesis of 17β-[4-(1,3-thiazoyl)]androstane 3β-hemisuccinate and glycoside
Drasar,Pouzar,Cerny,et al.
, p. 1039 - 1050 (2007/10/02)
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