243136-20-1Relevant academic research and scientific papers
Pilot-plant preparation of an αvβ3 integrin antagonist. Part 3. Process research and development of a diisopropylcarbodiimide and catalytic 1-hydroxybenzotriazole peptide coupling
, p. 1088 - 1093 (2009)
Studies directed toward the process research, development, and scale-up preparation of the potential αvβ3 integrin antagonist 1 are described. A convergent approach is detailed wherein tetrahydropyrimidine hydroxybenzoic acid 2 is li
