24558-42-7Relevant academic research and scientific papers
Hydroximoyl-tetrazole derivative fungicide
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Paragraph 0285; 0287; 0288, (2019/02/19)
The invention provides a hydroximoyl-tetrazole derivative fungicide, and particularly relates to hydroximoyl-tetrazole derivative, a preparing method thereof, application of hydroximoyl-tetrazole derivative serving as a fungicidal active agent, a form of
Amino sulfonyl compound, preparation method and uses thereof
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Paragraph 0186-0187, (2016/12/01)
The present invention relates to a new amino sulfonyl compound represented by a general formula I, or a tautomer, an enantiomer, a racemate or a pharmaceutically acceptable salt thereof, a preparation method, a pharmaceutical composition, and uses thereof, wherein the compound can be used for treatment of epilepsy, convulsion, obesity, and the like. The general formula I is defined in the specification.
IRE-1α INHIBITORS
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Paragraph 1369; 1370, (2016/10/07)
PROBLEM TO BE SOLVED: To provide compounds which directly inhibit inositol requiring enzyme 1 (IRE-1α activity) in vitro, prodrugs, and pharmaceutically acceptable salts thereof. SOLUTION: The present invention provides a compound represented by formula (A) [R3 and R4 are H or the like; Q5-Q8, together with the benzene ring to which they are attached, form a benzofused ring, where at least one of Q5-Q8 is a heteroatom selected from N, O, and S. COPYRIGHT: (C)2016,JPOandINPIT
Processes and intermediates for the preparation of N4-phenyl-quinazoline-4-amine derivatives
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Page/Page column 50, (2009/09/05)
This invention provides compounds of Formula (I), wherein B, G, A, E, R1, R2, R3, m and n are as defined herein, which are useful as type I receptor tyrosine kinase inhibitors, and methods of use thereof in the treatment of hyperproliferative disorders in mammals.
Benzisoxazole compounds useful as herbicides
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, (2008/06/13)
A herbicidal compound of formula (I): STR1 in which Ar is an optionally substituted aryl or heterocyclic ring system: R1 and R2 are independently selected from H, optionally substituted alkyl, alkenyl or akynyl, halogen, NRa Rb, or R1 and R2 together with the carbon to which they are attached form an optionally substituted alkenyl or cycloalkyl group; R3 is CO2 R4, CN, COR4, CH2 OR4, CH4 (OH)R4, CH(OR4)R5, CH2 OSO6 R4, CH2 OSO6 R4, CH2 ONR6 R7, CSNH2, COSR4, SCOR4, COHNSO2 R4, CONR6 R7, CONHNR6 R7, CONHN+ R6 R7 R8 Y-2, CO2- M+ or COON=CR6 R7 ; M+ is an agriculturally acceptable cation; Y- is an agriculturally acceptable anion; R4, and R5 are independently selected from H or an optionally substituted alkyl, aryl, alkenyl or alkynyl group; R6, R7, R8, R9, Ra and Rb are independently selected from H or an optionally substituted alkyl alkenyl, aryl or akynyl group or any two of R6, R7, R8, R9, Ra and Rb together with the atom to which they are attached form a cycloalkyl or heterocyclic ring; R6 and R7 may also be a heterocyclic ring; W is O or NR10 where R10 is H or lower alkyl; X is (CH2)n, CH=CH, CH(ORc)CH2, COCH2 ; where Rc is H or an optionally substituted alkyl, aryl, alkynyl or alkynyl group; and n is O, 1 or 2.
