2552-54-7

Usage

Uses

Used in Pharmaceutical Industry:
3-(Benzyloxy)isoxazole-5-carboxylic acid is used as a potential active pharmaceutical ingredient for its potential antimicrobial, anticancer, antiparasitic, and anti-inflammatory properties. Its isoxazole ring structure may contribute to its biological activities, making it a candidate for further research and development in drug discovery.
Used in Organic Synthesis:
3-(Benzyloxy)isoxazole-5-carboxylic acid is used as a synthetic intermediate in the preparation of various organic compounds. Its unique structure and potential reactivity may be exploited in the synthesis of complex molecules, including pharmaceuticals, agrochemicals, and other specialty chemicals.
Used in Research and Development:
3-(Benzyloxy)isoxazole-5-carboxylic acid is used as a research compound in academic and industrial laboratories. Its potential biological activities and structural features make it an interesting subject for studies aimed at understanding its properties, mechanisms of action, and potential applications in various fields, including medicine, materials science, and chemical engineering.

Upstream product

• 123320-44-5 (3-(benzyloxy)isoxazol-5-yl)methanol 
• 100-39-0 benzyl bromide 
• 205115-22-6 3-benzyloxyisoxazole-5-carboxylic acid methyl ester 
• 6567-35-7 3-bromo-5-isoxazolecarboxylic acid 
• 100-51-6 benzyl alcohol 

Downstream Products

• 104164-46-7 3-benzyloxy-5-isoxazolecarboxylic acid chloride 
• 2552-52-5 (3-benzyloxy-isoxazol-5-yl)-hydroxy-acetonitrile 
• 2552-51-4 (3-benzyloxy-isoxazol-5-yl)-hydroxy-acetic acid ethyl ester 
• 952318-51-3 C₁₂H₁₁NO₄S 
• 1252657-73-0 1-{[3-(Benzyloxy)isoxazol-5-yl]carbonyl}-4-(2-tert-butylphenyl)piperazine 
• 1198154-15-2 (3-benzyloxy-isoxazol-5-yl)-(2,3-dihydro-pyrido[4,3-b][1,4]oxazin-4-yl)-methanone 
• 916922-17-3 C₁₇H₁₃NO₄S 
• 104182-25-4 1-(3-benzyloxy-5-isoxazolyl)-2-bromoethanol 
• 104182-22-1 3-benzyloxy-5-bromoacetylisoxazole 
• 104164-47-8 3-benzyloxy-5-acetylisoxazole 
• 2552-53-6 3-benzyloxy-isoxazole-5-carbaldehyde 

Relevant academic research and scientific papers

Process Research and Development of an Enantiomerically Enriched Allyic Amine, One of the Key Intermediates for the Manufacture of Synthetic Tetracyclines

A robust, cost-effective, and high yielding manufacturing process for enantiomerically enriched (S)-allylic amine 3, a key intermediate for fully synthetic tetracyclines have been developed. Two novel and scalable asymmetric vinylations resulting in high-to-excellent stereoselectivity have been developed for the key step. The final product is purified by an efficient crystallization of a l-tartaric salt. The process described has been used to manufacture ～350 kg of the tartaric salt of 3 with 99.0% ee in 8 steps (35% overall yield) from cheap and readily available dimethyl maleate.

DERIVATIVES OF N-ACYL-N'-PHENYLPIPERAZINE USEFUL (INTER ALIA) FOR THE PROPHYLAXIS OR TREATMENT OF DIABETES

The present invention relates to a compound represented by the formula wherein each symbol is as defined in the present specification, which has a superior RBP4-lowering action and is useful as a pharmaceutical composition for the prophylaxis or treatment of a disease or condition mediated by an increase in RBP4.

ISOXAZOLE DERIVATIVE AND ISOTHIAZOLE DERIVATIVE HAVING INHIBITORY ACTIVITY ON 11 BETA -HYDROXYSTEROID DEHYDROGENASE TYPE I

Disclosed is a compound useful as an inhibitor of 11β-hydroxysteroid dehydrogenase type 1. A compound represented by the formula: a pharmaceutically acceptable salt or solvate thereof, wherein R1 is a group of the formula: -C(=O)NR4R

HETEROCYCLIC COMPOUND HAVING TYPE I 11 BETA HYDROXYSTEROID DEHYDROGENASE INHIBITORY ACTIVITY

Disclosed is a compound useful as a type I 11 β hydroxysteroid dehydrogenase inhibitor. A compound represented by the formula: a pharmaceutically acceptable salt or solvate thereof, wherein R1 is optionally substituted cycloalkyl, optionally su