259730-86-4Relevant academic research and scientific papers
Modeling directed design and biological evaluation of quinazolinones as non-peptidic growth hormone secretagogues
Ye, Zhixiong,Gao, Yingduo,Bakshi, Raman K.,Chen, Meng-Hsin,Rohrer, Susan P.,Feighner, Scott D.,Pong, Sheng-Shung,Howard, Andrew D.,Blake, Allan,Birzin, Elizabeth T.,Locco, Louis,Parmar, Rupa M.,Chan, Wanda W.-S.,Schaeffer, James M.,Smith, Roy G.,Patchett, Arthur A.,Nargund, Ravi P.
, p. 5 - 8 (2000)
Quinazolinone derivatives were synthesized and evaluated as non-peptidic growth hormone secretagogues. Modeling guided design of quinazolinone compound 21 led to a potency enhancement of greater than 200-fold compared to human growth hormone secretagogue affinity of a screening lead 4.
