28620-12-4Relevant articles and documents
Benzo[d]thiazol-2(3H)-ones as new potent selective CB2 agonists with anti-inflammatory properties
Leleu-Chavain, Natascha,Baudelet, Davy,Heloire, Valéria Moas,Rocha, Diana Escalante,Renault, Nicolas,Barczyk, Amélie,Djouina, Madjid,Body-Malapel, Mathilde,Carato, Pascal,Millet, Régis
, p. 347 - 362 (2019/01/04)
The high distribution of CB2 receptors in immune cells suggests their important role in the control of inflammation. Growing evidence offers this receptor as an attractive therapeutic target: selective CB2 agonists are able to modula
AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS
-
Page/Page column 99, (2016/11/17)
Provided herein are compounds of Formula (I), and pharmaceutically acceptable salts, N-oxides, or solvates thereof, [formula (I) should be inserted here]. Also provided herein are pharmaceutical compositions comprising compounds of Formula (I) and methods
Design and synthesis of 3-acyl-2(3H)-benzoxazolone and 3-acyl-2(3H)- benzothiazolone derivatives
Guenadil, Faouzi,Aichaoui, Hocine,Kapanda, Coco N.,Lambert, Didier M.,McCurdy, Christopher R.,Poupaert, Jacques H.
experimental part, p. 67 - 80 (2011/09/20)
A simpler and efficient "green" method using solid sodium hydroxide in a solvent mixture of acetone/water was found to catalyze N-acylation of 2(3H)-benzoxazolones and 2(3H)-benzothiazolones for facile and rapid synthesis of N-acyl derivatives in excellent yields. This method was applied to the synthesis of a series of 132 compounds employing a variety of acyl chlorides. Graphical abstract: [Figure not available: see fulltext.]
