291771-24-9Relevant academic research and scientific papers
Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1'-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1'-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines
Manfredini, Stefano,Lampronti, Ilaria,Vertuani, Silvia,Solaroli, Nicola,Recanatini, Maurizio,Bryan, David,Mckinney, Michael
, p. 1559 - 1566 (2007/10/03)
Few muscarinic antagonists differentiate between the M4 and M2 muscarinic receptors. In a structure-activity study, aimed at discovering leads for the development of a M4 muscarinic receptor-selective antagonist, we have s
