292820-10-1Relevant articles and documents
Bongkrekic Acid Analogue, Lacking One of the Carboxylic Groups of its Parent Compound, Shows Moderate but pH-insensitive Inhibitory Effects on the Mitochondrial ADP/ATP Carrier
Yamamoto, Atsushi,Hasui, Keisuke,Matsuo, Hiroshi,Okuda, Katsuhiro,Abe, Masato,Matsumoto, Kenji,Harada, Kazuki,Yoshimura, Yuya,Yamamoto, Takenori,Ohkura, Kazuto,Shindo, Mitsuru,Shinohara, Yasuo
, p. 1304 - 1322 (2015/10/28)
Bongkrekic acid, isolated from Burkholderia cocovenenans, is known to specifically inhibit the mitochondrial ADP/ATP carrier. However, the manner of its interaction with the carrier remains elusive. In this study, we tested the inhibitory effects of 17 bo
Macrocyclic diacylglycerol-bis-lactones as conformationally constrained analogues of diacylglycerol-lactones. Interactions with protein kinase C
Kang, Ji-Hye,Kim, Su Yeon,Lee, Jeewoo,Marquez, Victor E.,Lewin, Nancy E.,Pearce, Larry V.,Blumberg, Peter M.
, p. 4000 - 4007 (2007/10/03)
A series of macrocyclic diacylglycerol (DAG)-bis-lactones were investigated as extreme conformationally constrained analogues of DAG-lactones in order to seek more potent protein kinase C (PKC) ligands with higher binding affinities and less lipophilicity
