293733-51-4Relevant articles and documents
IMIDAZOPYRIDINONE COMPOUND
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Paragraph 0246, (2021/04/23)
The present invention aims to provide a novel compound which has prolyl hydroxylase (PHDs) inhibitory effect and which is useful for the treatment of inflammatory bowel diseases such as ulcerative colitis and the like. The present invention relates to a imidazopyridinone compound represented by the following formula (I) or a pharmaceutically acceptable salt thereof. The compounds of the present invention or pharmaceutically acceptable salts thereof which have prolyl hydroxylase inhibitory effect and, are useful as agents for the treatment of inflammatory bowel diseases such as ulcerative colitis and the like. In an embodiment, the present invention relates to a method for treating an inflammatory bowel disease
METHOD FOR PRODUCING IMIDAZOPYRIDINONE COMPOUND
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Paragraph 0218, (2021/09/27)
PROBLEM TO BE SOLVED: To provide a novel production method of an imidazopyridinone compound useful as a treatment agent for inflammatory bowel diseases (IBDs). SOLUTION: The present disclosure provides a method for the synthesis of, for example, an imidazopyridinone compound shown below. The method includes a process of introducing a desired substituent into the 1st-position of 2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridine, having an N-protected 3-pyrrolidino group at the 3rd-position; then deprotecting a 3rd-position substituent; and further introducing a desired substituent into N of the pyrrolidino group. SELECTED DRAWING: None COPYRIGHT: (C)2021,JPOandINPIT
SUBSTITUTED SULPHONAMIDES FOR CONTROLLING ANIMAL PESTS
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Paragraph 0346-0348, (2020/12/14)
The present invention relates to the use of a compound of the general formula (I) in which M and D have the meanings given in the description for controlling animal pests.