309757-83-3Relevant articles and documents
Synthesis, in vitro and in vivo biological evaluation, and comprehensive understanding of structure-activity relationships of dipeptidyl boronic acid proteasome inhibitors constructed from β-amino acids
Zhu, Yongqiang,Wu, Gang,Zhu, Xinrong,Ma, Yuheng,Zhao, Xin,Li, Yuejie,Yuan, Yunxia,Yang, Jie,Yu, Sen,Shao, Feng,Lei, Meng
supporting information; experimental part, p. 8619 - 8626 (2011/03/20)
An extensive structure-activity relationship (SAR) study of 72 dipeptidyl boronic acid proteasome inhibitors constructed fromβ -amino acids is reported. SAR analysis revealed that bicyclic groups at the R1 position, 3-F substituents at the Rsu
ARYLAMIDES
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Page/Page column 48, (2010/02/06)
The invention relates to compounds of formula (I), to a method for their production, to pharmaceutical compositions containing said compounds and to their use for the treatment and/or prophylaxis of human or animal diseases, in particular bacterial infections.
The asymmetric synthesis of β-haloaryl-β-amino acid derivatives
Bull,Davies,Delgado-Ballester,Fenton,Kelly,Smith
, p. 1257 - 1260 (2007/10/03)
Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.
