31052-85-4Relevant academic research and scientific papers
Might adrenergic α2C-agonists/α2A- antagonists become novel therapeutic tools for pain treatment with morphine?
Cardinaletti, Claudia,Mattioli, Laura,Ghelfi, Francesca,Del Bello, Fabio,Giannella, Mario,Bruzzone, Ariana,Paris, Hervé,Perfumi, Marina,Piergentili, Alessandro,Quaglia, Wilma,Pigini, Maria
experimental part, p. 7319 - 7322 (2010/09/07)
The imidazoline nucleus linked in position 2 via an oxyethylene bridge to a phenyl ring carrying an ortho substituent of moderate steric bulk provided α2-adrenergic (AR) ligands endowed with significant α2C- agonism/α2A-antagonism. S
